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取代芳甲酰哌嗪新衍生物的合成及其药理活性

SYNTHESIS AND POSITIVE INOTROPIC ACTIVITY OF SUBSTITUTED AROYL PIPERAZINE DERIVATIVES

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【作者】 徐鸣夏周国川杨艳谢益农刘智飞曾晓荣李瑞雪

【Author】 Xu Ming-Xia; Zhou Guo-Chuan; Yang Yan; Xie Yi-Nong ;Liu Zhi-Fei; Zeng Xiao-Rong; Li Rui-Xue ( School of pharmacy, West China University of Medical Sciences, Chengdu, 610041)( Luzhou Medical College, Luzhou, 646000) (3 Sichuan University, Chengdu, 61006

【机构】 华西医科大学药学院!成都610041沪州医学院!沪州646000四川大学!成都610064

【Abstract】 We designed and synthesized 5 new compounds. Their chemical structures were confirmed by means of MS, HNMR andelemental analysis. FPA was tested for positive inotropic activity. The results showed that FPA could increase the contrastive amplitudeof isolated atrium of guinea pigs and had no influence upon rhythm of the hearts.

  • 【文献出处】 化学研究与应用 ,CHEMICAL RESEARCH AND APPLICATION , 编辑部邮箱 ,1999年05期
  • 【分类号】TQ463.5
  • 【被引频次】4
  • 【下载频次】60
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