【摘要】 报道了一种铜/Selectfluor共催化的苄基碳氢键Ritter胺基化方法.该方法底物范围广泛,同时还具有高的区域选择性和化学选择性,避免使用强氧化剂和复杂的反应体系,在简单温和的反应条件下即可实现各种底物的苄基碳氢键胺基化.更多还原

【Abstract】 A copper/Selectfluor co-catalyzed Ritter-type benzylic C—H amination has been developed. The method has a wide substrate scope, and it also possesses high regioselectivity and chemoselectivity. It avoids the use of strong oxidants and complex reaction systems, enabling the amination of benzylic C—H bonds in various substrates under simple and mild reaction conditions.更多还原