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环溴虫酰胺(Cyclaniliprole)的合成与生物活性
Synthesis and Biological Activity of Cyclaniliprole
【摘要】 环溴虫酰胺(Cyclaniliprole)是日本石原产业公司开发的具双酰胺结构的新型广谱杀虫剂。为研究其合成方法与生物活性,以2-氨基-5-氯苯甲酸和3-溴-1-(3-氯-2-吡啶基)-1H-吡唑-5-羧酸为原料合成了环溴虫酰胺,并经质谱和核磁等确证了其结构。生物活性研究结果表明环溴虫酰胺(Cyclaniliprole)具有较好的杀虫活性。
【Abstract】 Cyclaniliprole is a novel broad-spectrum insecticide with diamide structure developed by Shihara Industry Co.,Ltd., Japan. In order to study the synthesis and biological activities, Cyclaniliprole was synthesized from2-amino-5-chlorobenzoic acid and 3-bromo-1-(3-chloro-2-pyridyl)-1 H-pyrazole-5-carboxylic acid. The structure was confirmed by MS and NMR etc. The results of bioassay showed that Cyclaniliprole exhibited good insecticidal activities.
【基金】 “十三·五”国家重点研发计划项目(2016YFD0300708)
- 【文献出处】 精细化工中间体 ,Fine Chemical Intermediates , 编辑部邮箱 ,2018年06期
- 【分类号】TQ453.2
- 【被引频次】4
- 【下载频次】233