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奥美沙坦酯的研究进展
Research Progress in Synthesis of Olmesartan Medoxomil
【摘要】 奥美沙坦是一种强效和特异性血管紧张素Ⅱ受体拮抗剂,用于治疗高血压,它的前体药物是奥美沙坦酯。介绍了奥美沙坦的药理作用,综述了奥美沙坦酯的合成方法,并对其市场前景作了展望。
【Abstract】 Olmesartan,a strongly effective and differential angiotensin Ⅱ receptor antagonist,is used to treat hypertensions.Its pro-drug is olmesartan medoxomil.In this paper,the mechanism was introduced,the synthetic methods were reviewed and the prospects were discussed.
【关键词】 奥美沙坦酯;
血管紧张素Ⅱ受体拮抗剂;
合成;
抗高血压药;
【Key words】 olmesartan medoxomil; angiotensin Ⅱ receptor antagonist; synthesis; antihypertensive drugs;
【Key words】 olmesartan medoxomil; angiotensin Ⅱ receptor antagonist; synthesis; antihypertensive drugs;
- 【文献出处】 化学与生物工程 , 编辑部邮箱 ,2005年04期
- 【分类号】R972.4
- 【被引频次】12
- 【下载频次】1272