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用Sn+2-树脂制备99m-Tc-平阳霉素

PREPARATION OF 99m-Te-PINGYANGMYCIN WITH Sn+2-RESIN

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【作者】 王鼎年; 李少林; 牟才宏; 向荣;

【Author】 Wang Dingnian, et alChongqing University of Medical Sciences, Chongqing.

【机构】 重庆医科大学基础核医学教研室; 重庆医科大学基础核医学教研室;

【摘要】 99m-Tc-平阳霉素是临床常用的亲肿瘤显影剂。用吸附Sn+2的阳离子交换树脂可以制得具有较好重复性的、稳定的99m-Tc-平阳霉素。标记率在90%以上。艾氏腹水实体癌小鼠分布实验表明99m-Tc-平阳霉素具有亲肿瘤作用。这种标记方法和其他方法比较,具有操作简便、可以作成药盒供临床使用等优点。

【Abstract】 99m-Tc-pingyangmycin (Bleomycin A5) has been widely used for clinical tumor ima-gingt Stannous ion adsorbed onto a cationic exchange resin shows specific characteristicsallowing the preparation of a stable 99m-Tc-pingyangmycin with good reproducibility.The labeling yeild is above 90%. The tumor-localization property of 99m-Tc-pingyangmycin was confirmed in mice inoculated with Ehrlich ascites tumor(solid form). Sn-resin labeling method has many advantages when compared with others, such as ease of performance and formulation of a Sn-resin kit system for clinical use.

【关键词】 99m-Tc-平阳霉素; 亚锡离子树脂; 肿瘤显影剂;
【Key words】 99m-Tc-pingyangmycin; stannous; ion; resin; tumor; imaging; agent;
  • 【文献出处】 重庆医药 ,Chongqing Medical Journal , 编辑部邮箱 ,1986年03期
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