【摘要】 “溃消净”,4-(3,4,5-三甲氧基硫代苯甲酰基)-四氢-1,4-氧嗪(商品名Trithiozine),在我们实验室试制成功。以没食子酸为原料,总收率达到57％。我们对此路线中的后面两个化合物进行了元素分析及光谱鉴定。“溃消净”的抑制胃酸分泌及抗溃疡作用可与甲氰咪胍(Cimetidine)相匹敌。更多还原

【Abstract】 "Kui Xiao Jing",4-(3,4,5-Trimethoxythiobenzoyl)-tetrahydro-1,4-oxazine (commercial name Trithiozine), has been synthesized in our laboratory. The total yield is 57％ from Gallic Acid. In this process, the two final products have been identified by elemental analysis and spectrum. Antisecretory and antiulcer effects of "Kui Xiao Jing" can be compared with those of "Cimetidine".更多还原